11-692 - Polypeptide Nanoparticles for Controlled Release of Ocular Biopharmaceuticals

Description:
  • Novel protein-based targeted drug delivery strategy
  • Potential application to treat several ocular disorders
  • Uses biocompatible, biodegradable and less immunogenic ELP-1 polymers

Abstract

USC scientists genetically engineered elastin-like polypeptides (ELP), which assemble multivalent nanoparticles at physiological temperature. The innovation was validated in a mouse model of age-related macular degeneration (AMD) with the intra-vitreal administration of aB crystallin. The ELP causes the therapeutic agent to be retained in the vitreous capsule where it can protect for at least 2 weeks.

Benefit

Market Application

Market Opportunity:

The delivery of drugs into the eye has always been a challenge, and so far, a general process hasn’t been discovered. Solutions are more specific to a certain type of drug or specific ocular disorder. Ocular injections are burdensome, and patient acceptance is a challenge. Additionally, low molecular weight peptides tend to be cleared rapidly from the ocular compartments, demanding repeated injections.

Hence there is a need for a versatile vehicle that reliably delivers the active ingredient into the eye, while being compatible with a variety of small molecule or biopharmaceutical drugs, and usable for different diseases.

Applications:

  • Therapeutic method for treating  ocular diseases
  • Intra-ocular drug delivery strategy

Publications

J Control Release. 2018 Aug 10; 283: 94–104.

Other

Stage of Development:

  • Tested in vitro and in vivo in mouse models
  • Available for exclusive and  non-exclusive license

Patent Information: